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Analysis and Application of Ligand Conformation in Drug Design
17 February 2016
Analysis and Application of Ligand Conformation in Drug Design

With the expertise of the team from C4X Discovery, this unique workshop will explore how conformational insights can impact rational design in drug discovery. The leaders will discuss the range of techniques available to experimentally determine molecular conformations, and their associated advantages and limitations. The case studies and discussion session will explore the principles of conformational design, and how such knowledge can be used to complement alternative design strategies and technologies.

Workshop LEADER

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Emma Blaney

Senior Programme Manager, C4X Discovery Limited

Emma Blaney, Senior Programme Manager, C4X Discovery


Dr Emma Blaney has been active in medicinal chemistry design since her PhD research at the University of Leeds. Since graduating in 2003 she has worked at GSK (Harlow) in Lead Optimisation and was more recently Section Head at Peakdale Molecular. Her ongoing interest in molecular design led her to join C4X Discovery as Senior Programme Manager. Her role is to lead the internal drug discovery programmes using the insights from the conformational design expertise of the company.
 

C4X Discovery Limited

C4X Discovery is a Manchester-based company focused on optimising drug discovery and design. The company uses its NMR-based technology to solve the dynamic 3D structures of a broad range of biomolecules. C4X Discovery's NMR technology shows what shapes active molecules prefer to adopt, providing high-quality templates for drug discovery and design. C4X Discovery is using its technology in collaboration with the pharmaceutical industry and to build its own proprietary pipeline of high-value therapeutic candidates.

Workshop agenda

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13:30

Registration

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14:00

Opening remarks and introductions

Emma Blaney, Senior Programme Manager, C4X Discovery Limited

Martin Watson, Head of NMR, C4X Discovery Limited

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14:10

Conformational design in drug discovery

- Introduction to molecular conformation

- Principles and objectives of conformational design

 

Emma Blaney, Senior Programme Manager, C4X Discovery Limited

Martin Watson, Head of NMR, C4X Discovery Limited

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14:50

C4X NMR analysis

- Outline of data collection and analysis

- Conformational model and descriptions

- Example structural analyses

 

Emma Blaney, Senior Programme Manager, C4X Discovery Limited

Martin Watson, Head of NMR, C4X Discovery Limited

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15:30

Afternoon Tea

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16:00

Case Studies and discussion session

- Interrogate how conformational insight can improve pharmacophore models

- Investigate how conformational design can improve selectivity profiles

 

Emma Blaney, Senior Programme Manager, C4X Discovery Limited

Martin Watson, Head of NMR, C4X Discovery Limited

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16:20

Topic Heading 8

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17:20

Closing remarks

Emma Blaney, Senior Programme Manager, C4X Discovery Limited

Martin Watson, Head of NMR, C4X Discovery Limited

VENUE

Holiday Inn Kensington Forum

97 Cromwell Road , London, United Kingdom

Holiday Inn Kensington Forum is perfectly situated in one of London’s most luxurious and beautiful areas within South Kensington. 

The hotel is just 2 minutes walk from Gloucester Road tube station for convenient travel to Hyde Park, London Eye, Tower Bridge plus more of London’s top attractions. There are also easy and direct links to some major transport hubs including Victoria, Kings Cross St Pancras, Paddington and Heathrow. 

This distinctive hotel in south London has so much to offer to make all guests really feel at home. The latest Holiday Inn relaunch is not just about the new look and feel for the hotel but to offer guests more benefits during their stay including a pillow menu for extra comfort during their sleep and a curved shower rail for more spacious feel. 

In addition to our 906 rooms, all business guests can take advantage of our meeting and conference facilities including High Speed Internet Access and unlimited Starbucks coffee at The Academy. Our hotel’s professional event planners are on board to help take the hard work and stress away from planning your next event. 

So whether you in London on business or pleasure, make the Holiday Inn London Kensington Forum your first choice of hotel and book your accommodation for our lowest internet rate guarantee. 

A number of our clients have been approached by third party organisations offering to book hotel rooms. We would advise that you do not book through them as they are not representing the SMi Group. SMi Group books all hotel rooms directly. If you are approached by a third party organisation then please contact us before making any bookings. If you have already booked a hotel room using a third party organisation, we would highly recommend contacting the hotel you were booked into to ensure a booking has been made for you. We would also advise you to please check the terms and conditions of the booking carefully.
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Holiday Inn Kensington Forum

97 Cromwell Road
London SW7 4DN
United Kingdom

Holiday Inn Kensington Forum

Holiday Inn Kensington Forum is perfectly situated in one of London’s most luxurious and beautiful areas within South Kensington. 

The hotel is just 2 minutes walk from Gloucester Road tube station for convenient travel to Hyde Park, London Eye, Tower Bridge plus more of London’s top attractions. There are also easy and direct links to some major transport hubs including Victoria, Kings Cross St Pancras, Paddington and Heathrow. 

This distinctive hotel in south London has so much to offer to make all guests really feel at home. The latest Holiday Inn relaunch is not just about the new look and feel for the hotel but to offer guests more benefits during their stay including a pillow menu for extra comfort during their sleep and a curved shower rail for more spacious feel. 

In addition to our 906 rooms, all business guests can take advantage of our meeting and conference facilities including High Speed Internet Access and unlimited Starbucks coffee at The Academy. Our hotel’s professional event planners are on board to help take the hard work and stress away from planning your next event. 

So whether you in London on business or pleasure, make the Holiday Inn London Kensington Forum your first choice of hotel and book your accommodation for our lowest internet rate guarantee. 

HOTEL BOOKING FORM

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WHAT IS CPD?

CPD stands for Continuing Professional Development’. It is essentially a philosophy, which maintains that in order to be effective, learning should be organised and structured. The most common definition is:

‘A commitment to structured skills and knowledge enhancement for Personal or Professional competence’

CPD is a common requirement of individual membership with professional bodies and Institutes. Increasingly, employers also expect their staff to undertake regular CPD activities.

Undertaken over a period of time, CPD ensures that educational qualifications do not become obsolete, and allows for best practice and professional standards to be upheld.

CPD can be undertaken through a variety of learning activities including instructor led training courses, seminars and conferences, e:learning modules or structured reading.

CPD AND PROFESSIONAL INSTITUTES

There are approximately 470 institutes in the UK across all industry sectors, with a collective membership of circa 4 million professionals, and they all expect their members to undertake CPD.

For some institutes undertaking CPD is mandatory e.g. accountancy and law, and linked to a licence to practice, for others it’s obligatory. By ensuring that their members undertake CPD, the professional bodies seek to ensure that professional standards, legislative awareness and ethical practices are maintained.

CPD Schemes often run over the period of a year and the institutes generally provide online tools for their members to record and reflect on their CPD activities.

TYPICAL CPD SCHEMES AND RECORDING OF CPD (CPD points and hours)

Professional bodies and Institutes CPD schemes are either structured as ‘Input’ or ‘Output’ based.

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The majority of Input and Output based schemes actively encourage individuals to seek appropriate CPD activities independently.

As a formal provider of CPD certified activities, SAE Media Group can provide an indication of the learning benefit gained and the typical completion. However, it is ultimately the responsibility of the delegate to evaluate their learning, and record it correctly in line with their professional body’s or employers requirements.

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